13
12
10
11
2
3
6
8
7
4
5
1
9
9
Fusion
CD4
Co-receptor (CCR5 or CXCR4)
Host Cell
Budding
Maturation
ALIX,ESCRT-I,ESCRT-III
Attachment
Env
HIV-1
Uncoating
Reverse
Transcription
NuclearExport
NuclearImport
Tat
Rev
Vpu
Vif
RNA Pol II
P-TEFb
Translation
Transcription
Release
AAA
AAA
AAA
AAA
AAA
AAA
AAA
AAA
AAA
5’LTR
3’LTR
IntegrationLEDGF
Accessory ViralProteins
Assembly
Pre-integration Complex
Gag
Gag
Pol
Translation
Gag
Gag
Pol
HIV Protease InhibitorsPepstatin ANelfinavirRitonavirLopinavir
Pan-CXCR AntagonistReparixinSelective-CXCR AntagonistsPlerixafor (CXCR4)SB225002 (CXCR2)WZ811 (CXCR4)
CCR AntagonistMaraviroc (CCR5)CCR AgonistZK756326 (CCR8)
Integrase InhibitorsRaltegravirDolutegravirElvitegravirCabotegravirBictegravir
Reverse TranscriptaseInhibitorsLamivudineEmtricitabineTenofovirZidovudineEfavirenz
CRM1 InhibitorsSelinexorEltanexorKPT-185Verdinexor
P
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Notes:
1:Clickable
2:Unclickable