Notes:
1:Clickable
2:Unclickable
SCF
Cbl
SFK
Shp2
Shc
Cbl
Grb2
Grb2
Grb2
Grb2
Cbl
BAD
Survival, Proliferation
Survival, Proliferation
Ubiquitination
PLCγ
Adhesion
Shp1
Shp2
Ubiquitination
APS
Lnk
SOCS6
P
P
P
P
P
P
P
P
c-Kit
PI3K
PI3K
JAK
Ras
Raf-1
MEK1/2
p38 MAPK
ERK
Akt
Akt
JAK2
STAT1
PLC
Pan-PI3K InhibitorsBEZ235GDC-0941LY294002Selective PI3K InhibitorsHS-173 (p110α)TGX-221 (p110β)CZC24832 (p110γ)CAL-101 (p110δ)
c-Kit InhibitorsMasitinibDovitinibAmuvatinibOSI-930Imatinib
Pan-JAK InhibitorsRuxolitinibMomelotinibAT9283Selective JAK InhibitorsAZD1480 (JAK2)Tofacitinib Citrate (JAK3)
Pan-Akt InhibitorsMK-2206PerifosineGSK690693Selective Akt InhibitorsA-674563 (Akt1)CCT128930 (Akt2)
Pan-MEK InhibitorsTrametinibU0126-EtOHPD184352Selective MEK InhibitorsSelumetinib (MEK1)BIX 02189 (MEK5)
Rho Family InhibitorsZoledronic AcidNSC 23766EHop-016ZCL278
ERK InhibitorsSCH772984XMD8-92FR 180204GDC-0994
Pan-p38 MAPK InhibitorsSB203580LY2228820VX-702LosmapimodSelective p38 MAPK InhibitorsBIRB 796 (p38α)Skepinone-L (p38α)
P
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