E
E
E
E
L
L
C
C
C
C
C
C
C
C
C
C
C
F
F
F
F
F
F
F
F
F
F
F
F
F
F
F
F
F
A
A
F
Kinase
Fibronetin
Cysteine Rich
Leucine Rich
EGF-Like
Acid Box
Cadherin
IG-Like
Glycine Rich
EGFR
HER2/ErbB2
ErbB3
ErbB4
INSR
IGF-1R
IRR
FGFR
PDGFR
CSF-1R
Kit
FLT3
VEGFR
Met
Ron
Sea
TrkA
TrkB
TrkC
Tie
Tie-2
Eph
Eck
Eek
Erk
Elk
Ros
Ret
Ltk
ALK
PLC
PDK-1
Akt
PKC
IKK
Syk
Bcr-Abl
Ras
Raf
c-Src
GSK-3
c-Jun
c-Fos
JAK
ROCK
Rho
PAK
JAK
STAT
PI3K/AktPathway
NF-κBPathway
MAPKPathway
Cell Cycle
JAK/STATPathway
Ⅰ
Ⅱ
Ⅲ
Ⅳ
Ⅴ
Ⅵ
Ⅶ
HER2/ErbB2 InhibitorsCP-724714AfatinibDacomitinib
Pan-EGFR InhibitorsAfatinibLapatinibSapitinibSelective EGFR InhibitorsErlotinib (EGFR/ErbB1)CP-724714 (HER2/ErbB2)Mutant EGFR InhibitorsOsimertinibGefitinib
Pan-FGFR InhibitorsBGJ398AZD4547ErdafitinibSelective FGFR InhibitorsPD173074 (FGFR1)H3B-6527 (FGFR4)
Pan-PDGFR InhibitorsImatinibCrenolanibCP-673451Selective PDGFR InhibitorsSunitinib (PDGFRβ)Avapritinib (PDGFRα)
c-Kit InhibitorsSitravatinibMasitinibAmuvatinibDovitinib
Pan-VEGFR InhibitorsAxitinibRegorafenibNintedanibLenvatinibSelective VEGFR InhibitorsCabozantinib (VEGFR2)Anlotinib (VEGFR2)SAR131675 (VEGFR3)
Tie-2 InhibitorsTie2 kinase InhibitorCabozantinib
c-RET InhibitorsAD80GSK3179106
ALK InhibitorsBrigatinibCeritinibLorlatinibAlectinibRepotrectinib
IGF-1R InhibitorsLinsitinibGSK1904529ABMS-754807Picropodophyllin
c-Met InhibitorsCrizotinib (PF-02341066)CapmatinibForetinib BMS-777607PHA-665752Savolitinib
Pan-Trk InhibitorsLarotrectinibEntrectinibSelitrectinibSelective Trk AntagonistANA-12 (TrkB)Selective Trk Agonist 7,8-Dihydroxyflavone (TrkB)
P
Cell Cycle
MAPK
Pathway
PI3K/Akt
Pathway
NF-κB
Pathway
JAK/STAT
Pathway
Kinase
Fibronetin
Cysteine Rich
Leucine Rich
EGF-Like
Acid Box
Cadherin
IG-Like
Glycine Rich
Tie
Eph
Eck
Eek
Erk
Elk
Ros
Ltk
Sea
IRR
I
II
III
IV
V
VI
VII
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Notes:
1:Clickable
2:Unclickable